
Galnon TFA
CAS No. 1217448-19-5
Galnon TFA ( —— )
产品货号. M37581 CAS No. 1217448-19-5
Galnon TFA 是一种选择性的非肽类的甘丙肽 GAL1 和 GAL2 受体激动剂,其 Ki 值分别为 11.7 和 34.1 μM。Galnon TFA 具有抗惊厥和抗焦虑作用。
纯度: >98% (HPLC)






规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥1034 | 有现货 |
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5MG | ¥1445 | 有现货 |
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10MG | ¥2196 | 有现货 |
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25MG | ¥3503 | 有现货 |
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50MG | ¥4927 | 有现货 |
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100MG | ¥6518 | 有现货 |
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200MG | ¥8645 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Galnon TFA
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Galnon TFA 是一种选择性的非肽类的甘丙肽 GAL1 和 GAL2 受体激动剂,其 Ki 值分别为 11.7 和 34.1 μM。Galnon TFA 具有抗惊厥和抗焦虑作用。
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产品描述Galnon TFA is a selective and non-peptide agonist of galanin GAL1 and GAL2 receptor, with Kis of 11.7 and 34.1 μM respectively. Galnon TFA exhibits anticonvulsant and anxiolytic effects.
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体外实验——
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体内实验——
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同义词——
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通路GPCR/G Protein
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靶点Neuropeptide Y Receptor
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受体Neuropeptide Y Receptor
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研究领域——
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适应症——
化学信息
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CAS Number1217448-19-5
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分子量792.84
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分子式C42H47F3N4O8
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纯度>98% (HPLC)
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溶解度In Vitro:?DMSO 中的溶解度 : 125 mg/mL (157.66 mM; 超声助溶 )
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SMILESC(C(O)=O)(F)(F)F.C(OC(N[C@@H](CC1CCCCC1)C(N[C@H](C(NC=2C=C3C(=CC2)C(C)=CC(=O)O3)=O)CCCCN)=O)=O)C4C=5C(C=6C4=CC=CC6)=CC=CC5
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献




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Neuropeptide Y (22-3...
Neuropeptide Y (22-36), a 15 amino acid peptide, is a fragment of Neuropeptide Y.Neuropeptide Y (NPY) is a 36 amino-acid neuropeptide that is involved in various physiological and homeostatic processes in both the central and peripheral nervous systems. NPY has been identified as the most abundant peptide present in the mammalian central nervous system, which consists of the brain and spinal cord. It is secreted alongside other neurotransmitters such as GABA and glutamate.
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L 152804
L 152804 是一种具有口服活性的、选择性的神经肽 Y Y5 受体 (NPY5-R) 拮抗剂,其对 hY5 的 Ki 值为 26 nM。L 152804 通过调节食物摄入和能量消耗,使饮食引起的肥胖小鼠体重减轻。
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Spexin
Potent galanin receptor 2/3 (GAL2/GAL3) agonist (EC50 values are 45.7 and 112.2 nM, respectively). Exhibits no significant activity at galanin receptor 1. Endogenous satiety-inducing peptide; inhibits long chain fatty acid uptake by adipocytes and decreases food consumption in diet-induced obese mice and rats. Attenuates LH secretion in goldfish. Exhibits anxiolytic effects in vivo.